Supply Rimegepant Supplier CAS 1289023-67-1

• Customization: Available
• CAS No.: 1289023-67-1
• Formula: 1289023-67-1
• Model NO.: Rimegepant
• Type: Pharmaceutical Intermediates
• Appearance: Powder
• Quality: Refined
• Colour: White
• Transport Package: Foil Bag
• Specification: 50g/100g/1kg/10kg/100kgs/1000kgs
• Trademark: MT
• Origin: China
• Production Capacity: 50/Month

Product Description

 

	Rimegepant
	[(5S,6S,9R)-5-amino-6-(2,3-difluorophenyl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-yl] 4-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxylate

Rimegepant (BMS-927711) (CGRP) ,Ki 0.027 nM.

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Ki: 0.027 nM (CGRP receptor)[1] IC50: 0.14 nM (CGRP receptor)[1]

Rimegepant(BMS-927711),CGRP,IC500.14±0.01 nM [1].

Rimegepant(BMS-927711),,CGRP[1].,Rimegepant(BMS-927711)(60,100300mg / kg)DBSAUC(0-24h)0.5-0.6.(DBS)Rimegepant[2].

:

DMSO:10 mg / mL(18.71 mM;)

:10 mg / mL(18.71 mM;)

:1.:90%PEG-300 10%:≥1mg / mL(1.87 mM);

1 mM	1.8707 mL	9.3535 mL	18.7070 mL
5 mM	0.3741 mL	1.8707 mL	3.7414 mL
10 mM	0.1871 mL	0.9353 mL	1.8707 mL

 

Contact Information

Mrs Dai